Compile Data Set for Download or QSAR
Found 33 of ic50 data for polymerid = 49000595,49000596
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50208989(CHEMBL506553)copy SMILEScopy InChI
Affinity DataIC50: 0.0790nMAssay Description:Displacement of [125I]galanin from human recombinant GAL1 receptor expressed in HEK293 cells measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)copy SMILEScopy InChI
Affinity DataIC50: 0.160nMAssay Description:Binding affinity to human GAL1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C5QPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)copy SMILEScopy InChI
Affinity DataIC50: 0.770nMAssay Description:Binding affinity to human GAL1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50149871((R)-2-((3-(biphenyl-4-yloxy)-3-(4-fluorophenyl)pro...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256665((3S,6S,9S,12S)-3-benzyl-9,12-di-sec-butyl-6-((2S,3...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256666((3S,6S,9S,12S)-3-benzyl-12-sec-butyl-6-((2S,3R)-3-...)copy SMILEScopy InChI
Affinity DataIC50: 10.2nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256705((3S,6S,9S,12S)-3-benzyl-6-((2S,3R)-3-hydroxybutan-...)copy SMILEScopy InChI
Affinity DataIC50: 11.1nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256704((3S,6S,9S,12S)-3-benzyl-9-sec-butyl-6-((2S,3R)-3-h...)copy SMILEScopy InChI
Affinity DataIC50: 11.4nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256664((S)-2-((2S,5S,8S,11S)-5-benzyl-8,11-di-sec-butyl-3...)copy SMILEScopy InChI
Affinity DataIC50: 20.4nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256706((3S,6S,9S,12S)-3-benzyl-6,9,12-tri-sec-butyl-1,4,7...)copy SMILEScopy InChI
Affinity DataIC50: 29.6nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256746((3S,6S,9S,15aR)-9-sec-butyl-6-((1-methoxy-1H-indol...)copy SMILEScopy InChI
Affinity DataIC50: 94.6nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ65WCPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358662(CHEMBL1922003)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358673(CHEMBL1922025)copy SMILEScopy InChI
Affinity DataIC50: 2.82E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358659(CHEMBL1922000)copy SMILEScopy InChI
Affinity DataIC50: 3.35E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358669(CHEMBL1922021)copy SMILEScopy InChI
Affinity DataIC50: 3.84E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358670(CHEMBL1922022)copy SMILEScopy InChI
Affinity DataIC50: 3.84E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358660(CHEMBL1922001)copy SMILEScopy InChI
Affinity DataIC50: 3.90E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358653(CHEMBL1921993)copy SMILEScopy InChI
Affinity DataIC50: 4.60E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358655(CHEMBL1921996)copy SMILEScopy InChI
Affinity DataIC50: 5.03E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358667(CHEMBL1922016)copy SMILEScopy InChI
Affinity DataIC50: 5.48E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358657(CHEMBL1921998)copy SMILEScopy InChI
Affinity DataIC50: 5.62E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358656(CHEMBL1921997)copy SMILEScopy InChI
Affinity DataIC50: 5.93E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358661(CHEMBL1922002)copy SMILEScopy InChI
Affinity DataIC50: 6.32E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358651(CHEMBL1921991)copy SMILEScopy InChI
Affinity DataIC50: 6.77E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358668(CHEMBL1922019)copy SMILEScopy InChI
Affinity DataIC50: 6.78E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358671(CHEMBL1922023)copy SMILEScopy InChI
Affinity DataIC50: 6.82E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358658(CHEMBL1921999)copy SMILEScopy InChI
Affinity DataIC50: 6.82E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358650(CHEMBL1921989)copy SMILEScopy InChI
Affinity DataIC50: 6.90E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358648(CHEMBL1921902)copy SMILEScopy InChI
Affinity DataIC50: 8.59E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358652(CHEMBL1921992)copy SMILEScopy InChI
Affinity DataIC50: 1.28E+4nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358672(CHEMBL1922024)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+4nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358654(CHEMBL1921995)copy SMILEScopy InChI
Affinity DataIC50: 2.75E+4nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358649(CHEMBL1921903)copy SMILEScopy InChI
Affinity DataIC50: 3.49E+4nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9QVTPubMed